Tapentadol

Tapentadol is an opioid pain reliever sold under the brand name, Nucynta. The forms of this analgesic are approved by various pharmaceutical regulation and certification agencies in countries across the globe, and considered highly effective.

Pain is an uncomfortable sensation that your nervous system uses to indicate that something may be wrong with your body. It can range from mild to moderate or can be more severe in some cases. For those receiving a medical diagnosis, pain is generally regarded as a symptom of an underlying medical condition. Pain may not always be curable, but it can be effectively managed with the use of analgesic medications.

Also available as a more potent painkiller, tapentadol 225 mg is formulated with 100 mg of the opioid pain medication and 125 mg of the muscle relaxer therapeutic, carisoprodol.

What is Tapentadol Used For?

• Tapentadol 50 mg is primarily used as a pain medication for both acute pain (pain that typically lasts for three to six months, or less) and chronic musculoskeletal pain (pain that normally lasts for longer than six months). This opioid painkiller is useful in managing the symptoms of moderate to severe pain as it functions in a similar manner to the dual action analgesic, tramadol, but is greater in efficacy than these pain tablets.
• The potency of this medication is somewhat in between the potency of tramadol and morphine, with analgesic effectiveness comparable to that of oxycodone.
• These pain-reliever tablets are also specifically formulated for the management of diabetic neuropathy (pain resulting from diabetes), especially when on-going treatment is required.

Tapentadol 50 mg Dosage

The 50 mg strength of this pain medicine is usually used for acute pain, that is, pain arising from injury or the discomfort that results from surgery.

This medication is available in immediate-release and extended-release formulations:

• Immediate-release: these pills release the therapeutic ingredients swiftly so that the analgesic effects may be experienced quickly. This form of the painkiller may be used for both acute and chronic pain relief.
• Extended-release: the extended-release form of Nucynta is generally useful for pain relief over a prolonged period of time as the active ingredient is released slowly. These formulations are not indicated for chronic pain relief.

Tapentadol 225 mg Dosage

Tapentadol 225 mg is a combination analgesic medication that is formulated with 100 mg Tapentadol and 125 mg carisoprodol. Carisoprodol is a musculoskeletal therapeutic which can be found under the trade name, Soma, among others.

This combination pain-reliever is available as the brand, Tofrodol-XX, and is suitable for severe pain, such as the neuropathy associated with diabetes.

Benefits of Tapentadol

Some of the benefits of Nucynta and Tofrodol-XX include:

• Greater efficacy: the medication is highly effective in relieving pain, more so than tramadol tablets. The combination analgesic of this opiate was specifically formulated to provide more efficacious analgesia.
• Less tolerance: opioids are generally known for their potential to cause tolerance when used in the long term. These pain-relievers have a lower potential to cause tolerance than other opioid pain medications.
• Less adverse effects: this pain therapeutic has a better side effect profile than other opiates.
• Can be used for neuropathic pain: the potency of these pain pills allow for them to be effective at relieving neuropathy. Research shows that chronic neuropathic patients have shown a better therapeutic response to tapentadol 225 mg than other opioid medicines.

Tapentadol vs Tramadol

Both these medications are opioid receptor agonists, meaning that they bind to the opioid receptors, and activate these, to bring forth their therapeutic benefits. However, tramadol has a binding affinity 6000 times less than Tofrodol-XX and in contrast, tapentadol 50 mg has been suggested to have 18 times less binding affinity than morphine. This is the reason why these opioid analgesics are thought to be in between the potency of tramadol and morphine.

In a study that compares the efficacy of tramadol and Nucynta in the treatment of low back pain, the latter pain medication was shown to be advantageous over the tramadol painkillers, in terms of pain control. This retrospective study was conducted on patients with musculoskeletal disorders, over a 24-week period, and reported tramadol as less superior in terms of analgesia (Guillen-Astete et. al., 2017). Although the latter option is considerably stronger, the milder opioid painkiller still has its place when treating cases of mild to moderate pain, even mildly severe pain in certain cases.

How Long do Tapentadol Effects Last?

This pain medication can last anywhere from four to six hours and the duration of action of these pills are very similar to that of carisoprodol, making for an ideal combination medication, as in the case of Tofrodol-XX.

The duration of action is, however, dependent, on several factors, such as age, gender, metabolism, body chemistry and so on, and these aspects all play a role in how long the therapeutic benefits of the medicine may last.

You can buy tapentadol 50 mg in extended-release form for prolonged therapeutic benefit.

Some Tapentadol Side Effects

As per the World Health Organisation (WHO), there is little evidence to indicate the potential risks of this medication. Although, according to clinical trials, the most frequently reported side effects associated with this analgesic were:

• Nausea
• Vomiting
• Dry mouth
• Headache
• Fatigue
• Itchiness

The side effects were mild to moderate in severity and were short-lived in most cases. However, if you are concerned about these adverse events, there are ways to effectively manage these symptoms.

Buy Tapentadol for Chronic Pain

As a more efficacious treatment for chronic pain, you can buy tapentadol 225 mg for the treatment of severe back pain, muscle injury, surgery pain and many other debilitating ailments.

Online pharmacies are particularly convenient for when you are unable to travel to a pharmacy because of the discomfort of pain symptoms, as these platforms only require a computer or smart phone and a stable internet connection.

You can buy tapentadol prescription free and paperless, through our safe and secure internet pharmacy. Expect rapid, discreet delivery matched with unrivalled service. There are customer service teams readily available to assist you with any enquiries or questions you may have regarding the service or the product you are purchasing. This leaves you with the peace of mind that you have chosen the best option to buy your medications.